3-aryl-7-chloro-3,4-dihydroacridine-1,9(2H,10H)-dione 1-oximes a

Details 3-aryl-7-chloro-3,4-dihydroacridine-1,9(2H,10H)-dione 1-oximes a 3-aryl-7-chloro-3,4-dihydroacridine-1,9(2H,10H)-dione 1-oximes a

1983-10-11

1986-06-03

Daus, Donald G.

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Heterocyclic carbon compounds containing a hetero ring...

514297, 544 59, 544162, 544361, 544363, 544392, 546103, 564 19, 564 36, 564250, A61K 31495, A61K 31435, C07D29504, C07D47100

Patent

active

045930279

ABSTRACT:
3-Aryl-7-chloro-3,4-dihydroacridine-1,9(2H,10H)-dione 1-oximes and 1-hydrazone derivatives of the formula I ##STR1## and their physiologically tolerated acid addition and ammonium salts are described, as is a process for their preparation. The new compounds are chemotherapeutic agents and are active against protozoa, especially malaria plasmodia.

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