Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Heterocyclic carbon compounds containing a hetero ring...
Patent
1984-06-26
1988-02-09
Daus, Donald G.
Drug, bio-affecting and body treating compositions
Designated organic active ingredient containing
Heterocyclic carbon compounds containing a hetero ring...
540573, A61K 3155, C07D24316
Patent
active
047242370
ABSTRACT:
Novel 2-substituted-aminomethyl-1,4-benzodiazepines which have been found to be antagonists of the function of cholecystokinins (CCK), to the preparation of these compounds, and to the use of these compounds to antagonize the function of CCK, which antagonism is useful, e.g., for the treatment and prevention of disorders of the gastrointestinal, central nervous and appetite regulatory systems of mammals, especially of humans.
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Bock Mark G.
Freidinger Roger M.
Abrams Samuel B.
Daus Donald G.
Elder Richard A.
Merck & Co. , Inc.
Pfeiffer Hesna J.
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