2-saccharinylmethyl aryl and aryloxy acetates useful as proteoly

Details 2-saccharinylmethyl aryl and aryloxy acetates useful as proteoly 2-saccharinylmethyl aryl and aryloxy acetates useful as proteoly

1994-08-08

1996-02-06

McKane, Joseph K.

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Having -c-, wherein x is chalcogen, bonded directly to...

548210, A61K 31425, C07D27506

Patent

active

054896045

ABSTRACT:
4-R.sup.4 -R.sup.5 -2-Saccharinylmethyl aryl and aryloxy acetates, useful in the treatment of degenerative diseases, are prepared by reacting a 4-R.sup.4 -R.sup.5 -2-halomethylsaccharin with an aryl or aryloxyacetic acid in the presence of an acid-acceptor.

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