2-saccharinylmethyl aryl and aryloxy acetates useful as proteoly

Details 2-saccharinylmethyl aryl and aryloxy acetates useful as proteoly 2-saccharinylmethyl aryl and aryloxy acetates useful as proteoly

1993-08-20

1995-01-31

Lee, Mary C.

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Having -c-, wherein x is chalcogen, bonded directly to...

5142315, 514254, 514321, 544135, 544368, 546198, 548210, 548211, C07D27504, A61K 31425

Patent

active

053859235

ABSTRACT:
4-R.sup.4 --R.sup.5 -2-Saccharinylmethyl aryl and aryloxy acetates, useful in the treatment of degenerative diseases, are prepared by reacting a 4-R.sup.4 --R.sup.5 -2-halomethylsaccharin with an aryl or aryloxyacetic acid in the presence of an acid-acceptor.

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