2-piperidones as intermediates for 5-deaza-10-oxo- and 5-deaza-1

Details 2-piperidones as intermediates for 5-deaza-10-oxo- and 5-deaza-1 2-piperidones as intermediates for 5-deaza-10-oxo- and 5-deaza-1

1991-12-20

1992-10-27

Tsang, Cecilia

Organic compounds -- part of the class 532-570 series

Organic compounds

Heterocyclic carbon compounds containing a hetero ring...

544279, C07F 702, C07D21136, C07D40100, A61K 31505

Patent

active

051590794

ABSTRACT:
4-Deaza-10-oxo- and 5-deaza-10-thio-5,6,7,8-tetrahydrofolic acid derivatives are provided as agents useful for treatment susceptible neoplasms in mammals. Pharmaceutical formulations and intermediates are also provided.

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