2-oxo-piperidinyl- and 2-oxo-azepanyl alkanoic acid...

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Heterocyclic carbon compounds containing a hetero ring...

Reexamination Certificate

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Details

C540S485000

Reexamination Certificate

active

07087596

ABSTRACT:
This invention relates to new 2-oxo-piperidinyl- and 2-oxo-azepanyl alkanoic acid derivatives of formula (1) having anticonvulsant activity which are useful as therapeutic agents for the treatment or prevention of epilepsy and other neurological disorders. The invention also concerns processes for preparing these derivatives and novel intermediates used in the preparation of these derivatives.

REFERENCES:
patent: 5334720 (1994-08-01), Schmiesing et al.
patent: 5719296 (1998-02-01), Acton, III et al.
patent: 5776950 (1998-07-01), Lee et al.
patent: 0 046 291 (1982-02-01), None
patent: 0 365 992 (1990-05-01), None
patent: 0 783 002 (1997-07-01), None
patent: 1 309 692 (1973-03-01), None
patent: 95 35308 (1995-12-01), None
patent: 01 19795 (2001-03-01), None
Piro, J. et al, Tetrahedron Letters, 42(5), pp. 871-873 (2001).
Estiarte, M.A. et al., Tetrahedron, 55(33), pp. 10173-10186 (1999).
Dutton, F.E. et al., Tetrahedron Letters, 39(30), pp. 5313-5316, (1998).
Robl, J.A. et al., Journal of Medicinal Chemistry, 39(2), pp. 494-502, (1996).
Robl, J.A. et al, J. Am. Chem. Soc., 116(6), pp. 2348-2355 (1994).
Depriest, S.A., et al, J. Am. Chem. Soc., 115(13), pp. 5372-5384 (1993).
De Laszlo, S.E. et al., J. Med. Chem., 35(5), pp. 833-846 (1992).
Aebi, J.D. et al., J. Med. Chem., 31(9), pp. 1805-1815 (1988).
Milewska M.J. et al., Synthesis, 12, pp. 1485-1488 (1996).
Prous, Drugs of the Future, 19(2), pp. 111-113 (1994).
Angelucci, L. et al., J. Med. Chem, 36(11), pp. 1511-1519 (1993).
Sreenivasan, U. et al., J. Med. Chem., 36(2), pp. 256-263 (1993).
Micouin L. et al., Tetrahedron, 52(22), pp. 7719-7726, (1996).

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