Drug – bio-affecting and body treating compositions – Antigen – epitope – or other immunospecific immunoeffector – Fungus – except allergen – or component thereof or substance...
Patent
1976-12-10
1979-06-12
Daus, Donald G.
Drug, bio-affecting and body treating compositions
Antigen, epitope, or other immunospecific immunoeffector
Fungus, except allergen, or component thereof or substance...
26032647, 542468, 546230, 546234, C07D20708, A61K 3140
Patent
active
041580605
ABSTRACT:
The invention provides novel 2-methoxy-benzamide derivatives of the formula: ##STR1## in which n is 1 or 2; R.sub.1 represents a cycloalkyl-alkyl radical of formula: ##STR2## a phenylalkyl radical of formula ##STR3## (in which m is an integer from 2 to 5, A is a linear or branched alkylene chain of 1 to 4 carbon atoms, and R.sub.4 is hydrogen, halogen, especially fluorine or chlorine, trifluoromethyl, or alkyl or alkoxy of 1 to 3 carbon atoms), CNCH.sub.2 --CH.sub.2 --, CH.tbd.C--CH.sub.2 --, ##STR4## R.sub.2 is either chlorine, SO.sub.2 R.sub.5 (in which R.sub.5 is alkyl of 1 to 4 carbon atoms), or SO.sub.2 NR.sub.6 R.sub.7 (in which, R.sub.6 and R.sub.7, which are identical or different, represent, independently of one another, hydrogen or alkyl of 1 to 4 carbon atoms); and R.sub.3 is hydrogen or alkyl of 1 to 4 carbon atoms; in the form of racemates or optical isomers, and their pharmaceutically acceptable acid addition salts, which are useful in the treatment of psychosomatic and psychotic disturbances.
REFERENCES:
patent: 3342826 (1967-09-01), Miller et al.
patent: 3723416 (1973-06-01), Thominet
patent: 3862139 (1975-01-01), Podesua et al.
patent: 3891671 (1975-06-01), Thominet
patent: 3923829 (1975-12-01), Denzler
patent: 3975434 (1976-08-01), Bulteau et al.
patent: 4021567 (1977-05-01), Kaplan et al.
patent: 4029673 (1977-06-01), Bulteau et al.
Giudicelli Don P. R. L.
Jalfre Maurice
Kaplan Jean-Pierre
Manoury Philippe M. J.
Najer Henry
Daus Donald G.
Lee Mary C.
Synthelabo
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