2-chloro and 2-bromo derivatives of 1,5-iminosugars

Details 2-chloro and 2-bromo derivatives of 1,5-iminosugars 2-chloro and 2-bromo derivatives of 1,5-iminosugars

1995-03-06

1997-03-18

Ivy, C. Warren

Organic compounds -- part of the class 532-570 series

Organic compounds

Four or more ring nitrogens in the bicyclo ring system

544224, 544242, 548110, 548125, 548126, 548146, 548152, 548215, 548217, 548251, 548406, 548517, 548518, 548519, 548541, 548556, C07F 702, C07D20700, C07D40500

Patent

active

056124805

ABSTRACT:
Novel 2-chloro and 2-bromo derivatives of 1,5-iminosugars are disclosed, especially such derivatives of 1,5-dideoxy-1,5-imino-D-glucitol. These compounds are useful inhibitors of glucosidase enzymes and also are useful as antiviral agents and as intermediates for the synthesis of other enzyme inhibitors and antiviral compounds.

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