2-chloro and 2-bromo derivatives of 1,5-iminosugars

Details 2-chloro and 2-bromo derivatives of 1,5-iminosugars 2-chloro and 2-bromo derivatives of 1,5-iminosugars

1996-06-14

1997-09-02

Ivy, C. Warren

Organic compounds -- part of the class 532-570 series

Organic compounds

Heterocyclic carbon compounds containing a hetero ring...

C07D21142

Patent

active

056633424

ABSTRACT:
Novel 2-chloro and 2-bromo derivatives of 1,5-iminosugars are disclosed, especially such derivatives of 1,5-dideoxy-1,5-imino-D-glucitol. These compounds are useful inhibitors of glucosidase enzymes and also are useful as antiviral agents and as intermediates for the synthesis of other enzyme inhibitors and antiviral compounds.

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