2,9-disubstituted purin-6-ones

Details 2,9-disubstituted purin-6-ones 2,9-disubstituted purin-6-ones

1996-01-12

1999-01-19

Berch, Mark L.

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Having -c-, wherein x is chalcogen, bonded directly to...

544265, A61K 3152, C07D47330, C07D23390

Patent

active

058614044

ABSTRACT:
2,9-Disubstituted purin-6-ones are prepared by acylating correspondingly substituted aminoimidazoles in a first step and then cyclizing the product to the purine. The new 2,9-disubstituted purin-6-ones can be employed as active compounds in medicaments, in particular for the treatment of inflammations, thromboembolic and cardiovascular diseases and diseases of the urogenital system.

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