Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Heterocyclic carbon compounds containing a hetero ring...
Patent
1989-06-08
1991-02-26
Rotman, Alan L.
Drug, bio-affecting and body treating compositions
Designated organic active ingredient containing
Heterocyclic carbon compounds containing a hetero ring...
5142268, 5142278, 514252, 514326, 514422, 546214, 546283, 544 60, 544152, 544374, 548517, C07D40512, C07D41312, A61K 3154, A61K 31495
Patent
active
049962035
ABSTRACT:
The present invention is directed to a specifically substituted tetrahydrofuran of the formula (I) ##STR1## wherein R.sup.4 is an alkylthio, alkylsulfinyl or alkylsulfonyl containing group and at least one of the substituents at positions 3,4 or 5 contains a heterocyclic, heteroaryl or substituted phenylthio moiety.
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Biftu Tesfaye
Bugianesi Robert L.
Girotra Nirindar N.
Kuo Chan H.
Ponpipom Mitree M.
DiPrima Joseph F.
Merck & Co. , Inc.
Panzer Curtis C.
Pfeiffer Hesna J.
Rotman Alan L.
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