Organic compounds -- part of the class 532-570 series – Organic compounds – Heterocyclic carbon compounds containing a hetero ring...
Patent
1998-10-01
2000-11-14
Kight, John
Organic compounds -- part of the class 532-570 series
Organic compounds
Heterocyclic carbon compounds containing a hetero ring...
548566, 548567, 548570, 548571, 548572, 549391, 549407, 549408, 549409, 549548, 549549, 549551, 549553, 549554, 549556, 549557, 549559, 549563, 560 14, 560 20, 560 21, 560 23, 560 24, 560102, 562433, 562434, 562462, 562466, 562469, 562492, 564164, 564165, 564166, 564167, 568307, 568325, 568327, 568440, 568441, 568442, 568592, 568661, 568705, 568715, 568808, C07D29500, C07D31180, C07D23300, C07D 4500, C07D30308
Patent
active
061472247
ABSTRACT:
Compounds of Formula 1, Formula 2 or Formula 3 where X is O, S, or (CR.sub.1 R.sub.1).sub.n where n is 0, 1 or 2; Y is a bivalent radical having Formula 4 or Formula 5 where o is an integer from 1 to 4 ##STR1## or Y is a bivalent aryl or 5 or 6 membered heteroaryl radical having 1 to 3 heteroatoms selected from N, S and O, said aryl or heteroaryl groups being unsubstituted, or substituted with 1 to 3 C.sub.1-6 alkyl or with 1 to 3 C.sub.1-6 fluoroalkyl groups; and the remaining symbols have the meaning described in the specification, have RXR selective retinoid agonist-like activity.
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Chandraratna Roshantha A.
Tsang Kwok Yin
Vasudevan Jayasree
Vuligonda Vidyasagar
Allergan Sales Inc.
Baran Robert J.
Covington Raymond
Kight John
Szekeres Gabor L.
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