1H-indazoles, benzothiazoles, 1,2-benzoisoxazoles,...

Details 1H-indazoles, benzothiazoles, 1,2-benzoisoxazoles,... 1H-indazoles, benzothiazoles, 1,2-benzoisoxazoles,...

2005-05-06

2009-12-15

Coleman, Brenda L (Department: 1624)

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Heterocyclic carbon compounds containing a hetero ring...

C540S556000

Reexamination Certificate

active

07632831

ABSTRACT:
The present invention relates generally to the field of ligands for nicotinic acetylcholine receptors (nAChR), activation of nAChRs, and the treatment of disease conditions associated with defective or malfunctioning nicotinic acetylcholine receptors, especially of the brain. Further, this invention relates to novel compounds (indazoles and benzothiazoles), which act as ligands for the α7 nAChR subtype, methods of preparing such compounds, compositions containing such compounds, and methods of use thereof.

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