1H-indazole-3-carboxamide-N-2-azabicyclo[2.2.2]octanes useful fo

Details 1H-indazole-3-carboxamide-N-2-azabicyclo[2.2.2]octanes useful fo 1H-indazole-3-carboxamide-N-2-azabicyclo[2.2.2]octanes useful fo

1989-10-03

1991-07-23

Rotman, Alan L.

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Having -c-, wherein x is chalcogen, bonded directly to...

546112, 514405, 548371, C07D40312, C07D45112, A61K 31445, A61K 31415

Patent

active

050343980

ABSTRACT:
Compounds of formula (I) and pharmaceutically acceptable salts thereof: ##STR1## wherein X is CO and Y is NH or O, or X is NH and Y is CO;

REFERENCES:
patent: 4886808 (1989-12-01), King
patent: 4937247 (1990-06-01), King
World Patents Index (Derwent), Accession No. 85-045742/08 (Feb. 1984).
Fludzinski et al., "Indazoles as Indole Bioisosteres: Synthesis and Evaluation of the Tropanoyl Ester and Amide of Indazole-3-carboxylate as Antagonists at the Serotonin 5-HT.sub.3 Receptor", J. Medicinal Chem., 30, pp. 1535-1537 (1987).
"5-HT.sub.3 Antagonists in Anxiety and Schizophrenia", SCRIP, No. 1246, Dec. 9, 1987, p. 23.

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