Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Having -c- – wherein x is chalcogen – bonded directly to...
Reexamination Certificate
2008-01-15
2008-01-15
Anderson, Rebecca (Department: 1626)
Drug, bio-affecting and body treating compositions
Designated organic active ingredient containing
Having -c-, wherein x is chalcogen, bonded directly to...
C548S262200
Reexamination Certificate
active
07319110
ABSTRACT:
The present invention relates to a group of 1H-1,2,4-triazole-3-carboxamide derivatives, to methods for the preparation of these compounds, and to pharmaceutical compositions containing at least one of these compounds as an active ingredient.These 1H-1,2,4-triazole-3-carboxamide derivatives are potent cannabinoid-CB1receptor agonists, partial agonists, inverse agonists or antagonists, useful for the treatment of disorders involving cannabinoid neurotransmission.The compounds have the general formula (I)wherein R and R1-R3have the meanings given in the specification.
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Kruse Cornelis G.
Lange Josephus H. M.
McCreary Andrew C.
Stuivenberg Herman H. van
Anderson Rebecca
Chung Susannah
Finnegan Henderson Farabow Garrett & Dunner L.L.P.
Solvay Pharmaceuticals B.V.
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