19-Nor-vitamin D compounds

Organic compounds -- part of the class 532-570 series – Organic compounds – 9,10-seco-cyclopentanohydrophenanthrene ring system or...

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556443, C07C40100

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active

056167440

ABSTRACT:
A 19-nor intermediate compound of the formula ##STR1## where R is the sidechain of a vitamin D derivative and where X.sub.1 and X.sub.2 are hydrogen or a hydroxy protecting group. The compounds are used in the preparation of 19-nor-vitamin D end products.

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Perlman, Kato et al, "1.alpha., 25-Dihydroxy-19-Nor-Vitamin D.sub.3, A Novel Vitamin D-Related Compound With Potential Therapeutic Activity" Tetrahedron Letters, vol. 31, No. 13, pp. 1823-1824, 1990.
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