17-ester, amide, and ketone derivatives of 3-oxo-4-azasteroids a

Details 17-ester, amide, and ketone derivatives of 3-oxo-4-azasteroids a 17-ester, amide, and ketone derivatives of 3-oxo-4-azasteroids a

1994-11-10

1996-04-23

Daus, Donald G.

Organic compounds -- part of the class 532-570 series

Organic compounds

Nitrogen attached directly or indirectly to the purine ring...

544405, 544406, 546 77, C07D24112, A61K 31495

Patent

active

055104851

ABSTRACT:
Described are new 17.beta.-ester, amide and ketone 4-aza-5a-androstan-3-ones and related compounds and their use as 5a-reductase inhibitors for treatment of benign prostatic hyperplasia and other hyperandrogenetic related disorders.

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