17.beta.-acyl-4-aza-5.alpha.-androst-1-ene-3-ones as 5.alpha. re

Details 17.beta.-acyl-4-aza-5.alpha.-androst-1-ene-3-ones as 5.alpha. re 17.beta.-acyl-4-aza-5.alpha.-androst-1-ene-3-ones as 5.alpha. re

1991-09-23

1992-09-29

Rivers, Diana G.

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Having -c-, wherein x is chalcogen, bonded directly to...

546 77, 514859, A61K 3158, C07J 7300

Patent

active

051514290

ABSTRACT:
17.beta.-Acyl-4-aza-5.alpha.-androst-1-en-3-ones of the formula: ##STR1## wherein R is selected from hydrogen, methyl and ethyl and

REFERENCES:
patent: 2227876 (1941-01-01), Bolt
patent: 3239417 (1966-03-01), DiTullio et al.
patent: 3264301 (1966-08-01), Doorenbos et al.
patent: 3285918 (1966-11-01), Doorenbos et al.
patent: 4220775 (1980-09-01), Rasmusson et al.
patent: 4377584 (1983-03-01), Rasmusson et al.
patent: 4732897 (1988-03-01), Cainelli et al.
patent: 4760071 (1988-07-01), Rasmusson et al.
patent: 4845104 (1989-07-01), Carlin et al.
patent: 4859681 (1989-08-01), Rasmusson et al.
Neri et al., Endo., vol. 91, No. 2, (1972), pp. 424-437.
Nayfeh et al., Steroids, 14, (1969), pp. 269-283.
Doorenbos & Solomon, J. Pharm. Sci., 62, 4, pp. 638-640 (1973).
Doorenbos & Brown, J. Pharm. Sci., 60, 8, pp. 1234-1235 (1971).
J. Org. Chem., vol. 46, No. 7, pp. 1442-1446, (Jul. 1981), by T. G. Back.
Chem. Abstracts, vol. 95, 109056j, by T. Liang et al. (1981).
JNCI, vol. 74, No. 2, pp. 475-481, Feb. 1985.
The Prostate, vol. 10, pp. 189-197, (1987), by G. L. Andriole et al.
J. Endocr., vol. 57, pp. 111-121, (1973), by K. D. Bingham et al.
Toxicol. Appl. Pharmacol., vol. 103, pp. 222-227, by G. L. Kedderis et al., (1990).
Doorebos & Kim, J. Pharm., 63, 4, pp. 620-622 (1974).
Rasmusson et al., J. Med. Chem., (1986), 29(11):2298-315.
Brooks et al., Prostate, (1986), 9(1):65-75.
Brooks et al., Steroids, (1986), 47(1):1-19.
Liang et al., Endocr., (1985), 117(2):571-579.
Rasmusson et al., J. Med. Chem., (1984), 27(12):1690-1701.

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