16-halogen-epothilone derivatives, process for their...

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Heterocyclic carbon compounds containing a hetero ring...

Reexamination Certificate

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Details

C514S183000, C540S454000, C540S462000

Reexamination Certificate

active

06930102

ABSTRACT:
A compund of formula I, an epothilone derivative, its method of preparation, and use as a pharmaceutical agent in treating malignant tumors

REFERENCES:
patent: 2004/0058969 (2004-03-01), Buchmann et al.
patent: 0 353 732 (1990-02-01), None
patent: 0 353 832 (1990-07-01), None
patent: 0 435 843 (1991-07-01), None
patent: WO 9825929 (1998-06-01), None
patent: WO-98/25929 (1998-06-01), None
patent: WO 9907692 (1999-02-01), None
patent: WO 0000485 (2000-01-01), None
CAPLUS Accession No: 2001:661399, abstract of “Synthesis of epothilones, intermediates, and analogs for use in treatment of cancers w/multidrug resistant phenotype,” PCT Int. Appl. No. WO 2001064650, Danishefshky et al (2001).
Crich, David et al: “Asymmetric synthesis of a taxol C-ring by aldol condensation and radical cyclization” TETAHEDRON (1977), 53 (21), 7127-7138, XP004105693; p. 7130.
Nagasawa, Kazuo et al: “An efficient asymmetric synthesis of 1.alpha., 25-(OH)2 vitamin D3 A-ring synthon” J. Org. Chem. (1993), 58(9), 2523-9, XP002150715; Seite 2524; Abbildung IV: Seite 2525; Abbildungen.
Allendinger, Thomas et al: “Fluoroolefin dipeptide isosteres. II. Enantioselective synthesis of both antipodes of the Phe-Gly Dipeptide mimic” Tetrahedron Lett. (1990), 31(50), 7301-4, Seite 7302.

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