13-Halo and 13-deoxy C-076 compounds

Details 13-Halo and 13-deoxy C-076 compounds 13-Halo and 13-deoxy C-076 compounds

1984-07-18

1985-10-15

Fan, Jane T.

Organic compounds -- part of the class 532-570 series

Organic compounds

Heterocyclic carbon compounds containing a hetero ring...

536 71, C07D49322

Patent

active

RE0320064

ABSTRACT:
Derivatives of the C-076 compounds are disclosed wherein the 13-position is unsubstituted or substituted by a halogen atom. The compounds are prepared by removing the glycosyl groups on the 13-position of the C-076 compounds isolated from the fermentation broth of Streptomyces avermitilis. This is followed by substitution of the 13-hydroxy group with a halogen, and subsequent removal of the halogen. The disclosed compounds are antiparasitic, anthelmintic, insecticidal and acaracidal agents.

REFERENCES:
patent: 3950360 (1976-04-01), Aoki et al.
Mishima et al., Tetrahedron Letters 10, pp. 711-714 1975.
Journal of Antibiotics 29(6), Jun. 1976, pp. 76-35 to 76-42 and pp. 76-14 to 76-16.
Derwent Abstract 76268w/46 to Sankyo Co.

Affiliated with

Also associated with

Rating

13-Halo and 13-deoxy C-076 compounds does not yet have a rating. At this time, there are no reviews or comments for this patent.

If you have personal experience with 13-Halo and 13-deoxy C-076 compounds, we encourage you to share that experience with our LandOfFree.com community. Your opinion is very important and 13-Halo and 13-deoxy C-076 compounds will most certainly appreciate the feedback.

Rate now

Comments { 0 }

Profile ID: LFUS-PAI-O-2430715