13-deoxy-23-imino derivatives of 13-deoxy C-076-aglycone compoun

Details 13-deoxy-23-imino derivatives of 13-deoxy C-076-aglycone compoun 13-deoxy-23-imino derivatives of 13-deoxy C-076-aglycone compoun

1987-08-27

1989-10-31

Raymond, Richard L.

Organic compounds -- part of the class 532-570 series

Organic compounds

Heterocyclic carbon compounds containing a hetero ring...

C07D31168

Patent

active

048778885

ABSTRACT:
The present invention relates to novel 23-imino derivatives of C-076 wherein the C-076 compounds are not substituted at the 13-position. The C-076 compounds (collectively) are isolates from the fermentation broth of Streptomyces avermitilis. The precursor 23-oxo compounds are prepared by selectively oxidizing suitably protected 13-deoxy C-076 aglycone compounds by using oxidizing agents. Subsequently, the 23-oxo compounds are converted to the 23-imino compounds. These novel compounds have potent anthelmintic, insecticidal, ectoparasticidal, nematicidal and acaricidal activity. Compositions containing these 23-oxo and 23-imino derivatives of 13-deoxy C-076 aglycones also are described herein.

REFERENCES:
patent: 4171314 (1979-10-01), Chabala et al.
patent: 4289760 (1981-09-01), Mrozik et al.
patent: 4423209 (1983-12-01), Mrozik
patent: 4427663 (1984-01-01), Mrozik
patent: 4457920 (1984-07-01), Mrozik
patent: 4547520 (1985-10-01), Ide et al.
Abstract of Japan 60/142991, Jul. 29, 1985.

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