11-substituted 5H,11H-pyrrolo(2,1-C) (1,4)benzoxazepines as anti

Details 11-substituted 5H,11H-pyrrolo(2,1-C) (1,4)benzoxazepines as anti 11-substituted 5H,11H-pyrrolo(2,1-C) (1,4)benzoxazepines as anti

1985-12-19

1987-05-19

Daus, Donald G.

Organic compounds -- part of the class 532-570 series

Organic compounds

Heterocyclic carbon compounds containing a hetero ring...

548518, C07D40106

Patent

active

046670394

ABSTRACT:
There are described to novel 11-substituted 5H,11H-pyrrolo[2,1-c][1,4]benzoxazepines of the general formula ##STR1## where m and n are each independently 0, 1 or 2 and m+n is 1 or 2, X and Y are each independently hydrogen, loweralkyl or halogen, and R is hydrogen, cyano, --C(NH.sub.2)NOH, ##STR2## unsubstituted loweralkyl, or substituted loweralkyl having one to three substituents each of which being independently cyano, hydroxy, cyclohexyl, furyl, thienyl, ##STR3## k being 1, 2 or 3, W being each independently hydrogen, halogen, hydroxy, loweralkyl, trifluoromethyl, loweralkoxy, nitro, amino, diloweralkylamino, phenoxy, or benzyloxy, and Z being hydrogen, loweralkyl or halogen, which are useful as antipsychotic and analgesic agents; novel intermediate compounds therefor; and methods of synthesizing the foregoing compounds.

REFERENCES:
patent: 3558652 (1971-12-01), Teotino et al.
patent: 3629435 (1971-01-01), Teotino et al.

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