Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Heterocyclic carbon compounds containing a hetero ring...
Patent
1990-06-29
1991-12-31
Scalzo, Catherine S. Kilby
Drug, bio-affecting and body treating compositions
Designated organic active ingredient containing
Heterocyclic carbon compounds containing a hetero ring...
544295, A61K 31505, C07D40300
Patent
active
050772937
ABSTRACT:
Certain 1-indolylalkyl-4-(alkoxypyrimidinyl)piperazines of Formula I are useful antidepressant agents. The ##STR1## substituents R.sup.1, R.sup.2 and R.sup.5 are hydrogen or lower alkyl; R.sup.3 and R.sup.4 are hydrogen, alkyl, alkoxy, alkythio, carboxamido, halo, or trifluoromethyl; R.sup.6 is alkoxy; and n is the integer 2 or 3.
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Mattson Ronald J.
Smith David W.
Yevich Joseph P.
Yocca Frank D.
Bristol-Myers Squibb Co.
Kilby Scalzo Catherine S.
Ryan Richard P.
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