1-arylsulphonyl, arylcarbonyl and arylthiocarbonyl pyridazino de

Details 1-arylsulphonyl, arylcarbonyl and arylthiocarbonyl pyridazino de 1-arylsulphonyl, arylcarbonyl and arylthiocarbonyl pyridazino de

1996-10-10

1998-05-19

Bernhardt, Emily

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Heterocyclic carbon compounds containing a hetero ring...

544234, A61K 3150, C07D23726, C07D49104, C07D49504

Patent

active

057536554

ABSTRACT:
1-Arylsulphonyl, arylcarbonyl and arylthiocarbonyl pyridazino derivatives and processes for making said derivatives are described. The novel derivatives are non-steroidal heterocyclic compounds which act as selective progestins and/or antiprogestins having a high in-vitro affinity for either the uterine, breast or bone progestin receptor. As such, the non-steroidal heterocyclic derivatives are useful in contraception, menopause, osteoporosis or endometriosis.

REFERENCES:
Advanced Organic Chemistry by Jerry March, pp. 382-384, 451-452 (1977).
Hogale et al, Chemical Abstracts, vol. 118, No. 213007 (1993).
Deshmurh et al, Chemical Abstracts, vol. 120, No. 323440 (1994).
McGuire et al, Biochemistry, vol. 13, pp. 319-322 (1974).
Holava et al, J. Med. Chem. 14, pp. 262-264 (1971).
Aubagnac et al, Bull. Chem. Soc. France pp. 2859-2868 (1972).

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