1-aroyl-3-indolyl alkanoic acids and derivatives thereof useful

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Having -c- – wherein x is chalcogen – bonded directly to...

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514419, 548500, A61K 3140, A61K 31405, C07D20912

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active

054362652

ABSTRACT:
Compounds of the structures shown below are specific inhibitors of cyclooxygenase-2 useful in the treatment of cyclooxygenase-2 mediated disease states such as inflammation, pain and fever, and are non-ulcerogenic. ##STR1##

REFERENCES:
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patent: 3647858 (1972-03-01), Hinkley et al.
patent: 3654349 (1972-04-01), Shen et al.
patent: 4868201 (1989-09-01), Fukaya et al.
Chemical Abstracts vol. 106:50037v, 1987, Fukaya et al, "Indoleacetic Acid Derivatives."
Chemical Abstracts vol. 91:102002y, 1979, Stochla et al, "Antiinflammatory activity of . . . in immunological and non-immunological tests".
Chemical Abstracts vol. 64, 1966, Abstract 6622b, ".alpha.-1 (Aroyl-3-indolyl)acetic Acids".
Chemical Abstracts vol. 59, 1963, abstract 8707e, "Indoles."
Chemical Abstracts, vol. 62, 1965, abstract 16198e, "Indole acid Amides."
Advances in Drug Research, vol. 12, 1977 p. 145, Harper, N. J. et al, New York.
Agnew. Chem. Internat. Edit. vol. 11 (1972) No. 6 pp. 460-472, "Perspectives in Nonsteroidal Anti-Inflammatory Agents", T. Y. Shen.
Arzneim.Forsch. Drug Res. 30 (II), Nr. 8a (1980) Boltze, et al. pp. 1314-1325.

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