1-alkyl-4-(3-substitutedphenyl)piperidines

Details 1-alkyl-4-(3-substitutedphenyl)piperidines 1-alkyl-4-(3-substitutedphenyl)piperidines

2007-09-04

2007-09-04

Desai, Rita (Department: 1625)

Organic compounds -- part of the class 532-570 series

Organic compounds

Heterocyclic carbon compounds containing a hetero ring...

C546S229000, C546S237000

Reexamination Certificate

active

10987527

ABSTRACT:
8-Substituted-2,6-methano-3-benzazocines of general structure I in which A is —CH2—OH, —CH2NH2, —NHSO2CH3,and Y is O, S orNOH are useful as analgesics, anti-diarrheal agents, anticonvulsants, antitussives and anti-addiction medications.8-Carboxamides, thiocarboxamides, hydroxyamidines and formamides are preferred.

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