Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Having -c- – wherein x is chalcogen – bonded directly to...
Reexamination Certificate
2011-06-28
2011-06-28
Kosack, Joseph R (Department: 1626)
Drug, bio-affecting and body treating compositions
Designated organic active ingredient containing
Having -c-, wherein x is chalcogen, bonded directly to...
C514S422000, C514S361000, C514S343000, C514S414000, C514S326000, C514S254010, C514S237200, C514S399000, C514S218000, C514S316000, C514S217080, C514S227800, C514S292000, C548S127000, C548S518000, C548S527000, C548S537000, C548S530000, C548S467000, C548S314700, C540S575000, C540S602000, C544S060000, C544S141000, C546S087000, C546S187000, C546S208000, C546S279100
Reexamination Certificate
active
07968591
ABSTRACT:
1,3-disubstituted 4-methyl-1H-pyrrole-2-carboxamides corresponding to formula Imethods for their production, pharmaceutical compositions containing them, and the use thereof for noradrenalin receptor regulation, particularly for inhibiting noradrenalin reuptake, and/or for 5-HT receptor regulation, particularly for inhibiting 5-hydroxy tryptophan reuptake, and/or for opioid receptor regulation and/or for batrachotoxin (BTX) receptor regulation and/or for treating or inhibiting pain and other conditions.
REFERENCES:
patent: 5189055 (1993-02-01), Thal et al.
patent: 5698581 (1997-12-01), Kleemann et al.
patent: 7250443 (2007-07-01), Desai et al.
patent: 2005/0014765 (2005-01-01), Mailliet et al.
patent: 2007/0135494 (2007-06-01), Merla et al.
patent: 0 957 099 (1999-11-01), None
patent: WO 90/02733 (1990-03-01), None
patent: WO 2004/018455 (2004-03-01), None
patent: WO 2004/108685 (2004-12-01), None
patent: WO 2005/113497 (2005-12-01), None
Alazard et al. Bulletin de la Societe Chimique de France, 1993, 130, 779-87.
Registry Database for Registry No. 172458-72-9, entered STN on Jan. 19, 1996.
Alazard, J.P., et al., “Composés interagissant avec la tubuline. Partie I: synthèse de phénylpyrrolesortho-ortho' substitués en rotation libre ou empêchée”, Bull. Soc. Chim. Fr., 1993, vol. 130, No. 6, pp. 779-787. XP009090907.
German Search Report dated Dec. 19, 2006 including portions translated in English (Eight (8) pages).
International Search Report dated Oct. 22, 2007 including portion translated in English (Seven (7) pages).
PCT/ISA/237 including English translation (Nine (9) pages), Jan. 12, 2009.
Bijsterveld Edward
Hennies Hagen-Heinrich
Oberboersch Stefan
Sundermann Bernd
Sundermann Corinna
Coughlin Matthew P
Crowell & Moring LLP
Gruenenthal GmbH
Kosack Joseph R
LandOfFree
1,3-disubstituted 4-methyl-1H-pyrrole-2-carboxamides and... does not yet have a rating. At this time, there are no reviews or comments for this patent.
If you have personal experience with 1,3-disubstituted 4-methyl-1H-pyrrole-2-carboxamides and..., we encourage you to share that experience with our LandOfFree.com community. Your opinion is very important and 1,3-disubstituted 4-methyl-1H-pyrrole-2-carboxamides and... will most certainly appreciate the feedback.
Profile ID: LFUS-PAI-O-2738110