1,3-/1,4-thiomorpholino-terminated non-peptidyl .alpha.-succinam

Details 1,3-/1,4-thiomorpholino-terminated non-peptidyl .alpha.-succinam 1,3-/1,4-thiomorpholino-terminated non-peptidyl .alpha.-succinam

1993-12-16

1995-06-13

Brust, Joseph Paul

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Heterocyclic carbon compounds containing a hetero ring...

5142272, 5142275, 544 54, 544 584, A61K 3154, C07D27906, C07D27912

Patent

active

054243076

ABSTRACT:
Non-peptidyl compounds characterized generally as .alpha.-succinamidoacyl aminodiols having a 1,3-thiomorpholino-type group or a 1,4-thiomorpholino-type group at the N-terminus are useful as renin inhibitors for the treatment of hypertension.

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