1,2-dihydroquinoline derivative having (substituted phenyl...

Details 1,2-dihydroquinoline derivative having (substituted phenyl... 1,2-dihydroquinoline derivative having (substituted phenyl...

2011-08-30

2011-08-30

Seaman, D (Department: 1625)

Organic compounds -- part of the class 532-570 series

Organic compounds

Heterocyclic carbon compounds containing a hetero ring...

C546S167000, C546S180000

Reexamination Certificate

active

08008497

ABSTRACT:
The compounds represented in general formula (1) and a salt thereof are useful for glucocorticoid receptor modulator.The R1represents a hydrogen atom or a lower alkyl group; R2represents a hydrogen atom or a lower alkyl group; R3and R4may be the same or different and represent a hydrogen atom or a lower alkyl group; R5represents a hydrogen atom or a lower alkyl group; R6represents a halogen atom, a lower alkyl group, a hydroxy group, a lower alkoxy group, a nitro group or a cyano group; X represents —C(O)—, —C(O)NR8—, —S(O)2— and the like; R7and/or R8may be the same or different and represent a hydrogen atom, a lower alkyl group which may have a substituent, an aryl group which may have a substituent, a heterocyclic group which may have a substituent, a lower alkoxy group which may have a substituent and the like; Y represents a lower alkylene group; Z represents a benzene ring or a heterocyclic ring; and P represents 0, 1, 2 or 3.

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