1,2-dihydroquinoline derivative having substituted...

Details 1,2-dihydroquinoline derivative having substituted... 1,2-dihydroquinoline derivative having substituted...

2011-08-30

2011-08-30

Seaman, D (Department: 1625)

Organic compounds -- part of the class 532-570 series

Organic compounds

Heterocyclic carbon compounds containing a hetero ring...

C546S167000, C546S180000

Reexamination Certificate

active

08008496

ABSTRACT:
The compounds represented in general formula (1) and a salt thereof are useful for glucocorticoid receptor modulator.The R1represents a hydrogen atom or a lower alkyl group; R2represents a hydrogen atom or a lower alkyl group; R3and R4may be the same or different and represent a hydrogen atom or a lower alkyl group; R5represents a hydrogen atom or a lower alkyl group; R6represents a halogen atom, a lower alkyl group, a hydroxy group, a lower alkoxy group or a nitro group; X represents —C(O)—, —C(O)NR8—, —S(O)2— and the like; R7and/or R8may be the same or different and represent a hydrogen atom, a lower alkyl group which may have a substituent, an aryl group which may have a substituent, a heterocyclic group which may have a substituent, a lower alkoxy group which may have a substituent and the like; Y represents a lower alkylene group; Z represents a chalcogen atom; and P represents 0, 1, 2 or 3.

REFERENCES:
patent: 5688808 (1997-11-01), Jones et al.
patent: 5688810 (1997-11-01), Jones et al.
patent: 6852719 (2005-02-01), Liu et al.
patent: 2004/0116455 (2004-06-01), Bekkali et al.
patent: 2007/0254917 (2007-11-01), Higuchi et al.
patent: 2009/0298826 (2009-12-01), Matsuda et al.
patent: 2009/0298827 (2009-12-01), Matsuda et al.
patent: 2009/0326009 (2009-12-01), Matsuda et al.
patent: 1 944 290 (2008-07-01), None
patent: 10-510840 (1998-10-01), None
patent: 2002-193955 (2002-07-01), None
patent: WO 96/19458 (1996-06-01), None
patent: WO 96/19458 (1996-06-01), None
patent: WO 2004/018429 (2004-03-01), None
patent: WO 2006/019716 (2006-02-01), None
patent: WO 2007/032556 (2007-03-01), None
patent: 2008/111632 (2008-09-01), None
patent: WO 2008/111632 (2008-09-01), None
Supplementary European Search Report dated Nov. 4, 2010 in European Patent Application No. 07 83 1811.
Hajime Nawata, Sougou Rinsyou, “New horizon of glucocorticoid therapy in 21stcentury,” 54(7), pp. 1951-2076 (2005).
Ku, Yi-Yin; Grieme, et al., “Asymmetric Synthesis of A-240610.0 via a new Atropselective Approach for Axially Chiral Biaryls with Chirality transfer,” Journal of the American Chemical Society, vol. 124, 2002, pp. 4282-4286.
U.S. Appl. No. 11/992,088, filed Mar. 14, 2008, Confirmation No. 4161.
Sougou Rinsyou, 54(7), 1951-2076 (2005) and English translation of identified portions of pp. 1952-2073.
U.S. Appl. No. 12/312,393, filed May 7, 2009, Confirmation No. 6179.
U.S. Appl. No. 12/312,396, filed May 7, 2009, Confirmation No. 5788.

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