1,2,5,6-tetrahydropyridyl triazoles and tetrazoles useful as fun

Details 1,2,5,6-tetrahydropyridyl triazoles and tetrazoles useful as fun 1,2,5,6-tetrahydropyridyl triazoles and tetrazoles useful as fun

1987-12-01

1989-11-28

Lee, Mary C.

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Having -c-, wherein x is chalcogen, bonded directly to...

548558, 548561, 514427, A61K 3140, C07D20750, C07D207337

Patent

active

048838071

ABSTRACT:
Compounds of the formula (I): ##STR1## and stereoisomers and salts thereof, wherein R.sup.1 and R.sup.2, are optionally substituted alkyl; V is either oxygen or sulphur; Y is hydrogen, optionally substituted alkyl, cyano, nitro or halogen; X is ##STR2## Z is NOR.sup.5 or ##STR3## A is CO.sub.2 R.sup.6, COR.sup.7, cyano, nitro or acylamino; B is hydrogen, optionally substituted alkyl, optionally substituted aryl, CO.sub.2 R.sup.8, COR.sup.9, cyano, nitro or acylamino, or A and B together form a ring containing one or more heteroatoms; R.sup.4 is CO.sub.2 R.sup.3 or R.sup.17 ; R.sup.12 is OR.sup.13, SR.sup.14, NR.sup.15 R.sup.16 or R.sup.18 ; R.sup.3 is optionally substituted alkyl;and R.sup.5 to R.sup.11 and R.sup.13 to R.sub.18, which are the same or different, are hydrogen, optionally substituted alkyl, optionally substituted cycloalkyl, optionally substituted cycloalkylalkyl, optionally substituted alkenyl, optionally substituted alkynyl, optionally substituted aralkyl, optionally substituted aryl, or optionally substituted heteroaryl, or R.sup.10 and R.sup.11, or R.sup.15 and R.sup.16 together with their adjacent nitrogen atom join to form a saturated ring (except that R.sup.10 and R.sup.11, together with their adjacent nitrogen atom, do not form an unsubstituted piperidine ring when R.sup.1 and R.sup.2 are both methyl, Y is hydrogen and V is oxygen) optionally containing one or more hetero atoms in addition to the nitrogen atom, for example, a pyrrolidine or morpholine. These compounds are useful in agriculture, for example, as fungicides or plant growth regulators.

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