Pyrazolobenzazepines

Details Pyrazolobenzazepines Pyrazolobenzazepines

1981-07-23

1983-04-12

Rollins, Alton D.

Chemistry of carbon compounds

Miscellaneous organic carbon compounds

C-metal

260465G, 260465K, 424273P, 548378, 562435, 562436, 562460, 562491, 564328, 568424, 568425, 568705, 568809, A61K 3155, C07D48704

Patent

active

043797652

ABSTRACT:
There are presented compounds of the formulas ##STR1## wherein R.sub.1 is hydrogen or lower alkyl; R.sub.2 and R.sub.3 are selected from the group consisting of hydrogen, lower alkyl, C.sub.2 to C.sub.7 carboxylic acids, hydroxy C.sub.2 to C.sub.7 alkyl, C.sub.2 to C.sub.7 carboxylic acid esters and amides and the group COR.sub.11 wherein R.sub.11 is alkoxy, amino or mono- lower alkyl amino; R.sub.6 is nitro or halo and R.sub.5 is hydrogen or halo,
and the pharmaceutically acceptable salts thereof.
The pyrazolobenzazepines are useful as anxiolytic and sedative agents.
Also provided are processes and intermediates in the production of the above pyrazolobenzazepines.

REFERENCES:
patent: 4028381 (1977-06-01), Gschwend

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