Carbostyril derivatives, process for producing the same and card

Details Carbostyril derivatives, process for producing the same and card Carbostyril derivatives, process for producing the same and card

1983-08-22

1984-08-28

Daus, Donald G.

Drug, bio-affecting and body treating compositions

Antigen, epitope, or other immunospecific immunoeffector

Bacterium or component thereof or substance produced by said...

546157, 546158, 544128, 544363, 4242484, 424250, C07D21520, A61K 3147

Patent

active

044684029

ABSTRACT:
Novel carbostyril derivatives and their pharmaceutically acceptable salts represented by the formula (I) ##STR1## wherein R.sup.1 is a hydrogen atom, a lower alkyl group, a lower alkenyl group, a lower alkynyl group or a phenyl-lower alkyl group; R.sup.2 and R.sup.3 may be the same or different and each is a lower alkyl group which may have one hydroxy group or one halogen atom as the substituent, or a phenyl-lower alkyl group which may have 1 to 3 substituents selected from the group consisting of a lower alkoxy group and a halogen atom on the phenyl ring, or said phenyl-lower allkyl group may have a lower alkylenedioxy group as the substituent on the phenyl ring; further R.sup.2 and R.sup.3 may form, together with the adjacent nitrogen and without an additional hetero-atom, a 5-or 6 membered saturated heterocyclic ring which may have a lower alkyl group or a phenyl-lower alkyl group as the substituent; the carbon-carbon bond between 3- and 4-positions in the carbostyril skeleton being a single or double bond. The derivatives are useful as the active ingredient in cardiotonic compositions.

REFERENCES:
patent: 3555030 (1971-01-01), Loev et al.
patent: 3994900 (1976-11-01), Krapcho et al.
patent: 4022776 (1977-05-01), Nakagawa et al.
patent: 4022784 (1977-05-01), Nakagawa et al.
patent: 4070470 (1978-01-01), Nakagawa et al.
patent: 4210753 (1980-07-01), Tominaga et al.
patent: 4223137 (1980-09-01), Yoshizaki et al.
patent: 4256890 (1981-03-01), Nakagawa et al.
patent: 4298739 (1981-11-01), Nishi et al.

Affiliated with

Also associated with

Rating

Carbostyril derivatives, process for producing the same and card does not yet have a rating. At this time, there are no reviews or comments for this patent.

If you have personal experience with Carbostyril derivatives, process for producing the same and card, we encourage you to share that experience with our LandOfFree.com community. Your opinion is very important and Carbostyril derivatives, process for producing the same and card will most certainly appreciate the feedback.

Rate now

Comments { 0 }

Profile ID: LFUS-PAI-O-877250