Stereocontrolled acetoxyazetidinone process

Details Stereocontrolled acetoxyazetidinone process Stereocontrolled acetoxyazetidinone process

1986-01-13

1987-01-27

Rizzo, Nicholas S.

Organic compounds -- part of the class 532-570 series

Organic compounds

Heterocyclic carbon compounds containing a hetero ring...

540357, C07D49900, A61K 31425

Patent

active

046393358

ABSTRACT:
A novel stereocontrolled process is disclosed for converting 6-aminopenicillanic acid to an optically active azetidinone of the formula ##STR1## wherein R" is a hydroxy-protecting group by use of a 6,6-dihaloanhydropenicillin or 6,6-bis(phenylselenyl)anhydropenicillin intermediate.

REFERENCES:
patent: 4468351 (1984-08-01), Pirie et al.
Heterocycles 17: 201-207 (1982) Hirai et al., J. Org. Chem. 42: 2960-2965 (1977) DiNinno et al.
Tetrahedron Letters 23(39): 4021-4024 (1982) Hirai et al.
Tetrahedron Letters 23(22): 2293-2296 (1982) Reider et al.
Chem. Pharm. Bull 29(11): 3158-3172 (1981) Hayashi et al.

Affiliated with

Also associated with

Rating

Stereocontrolled acetoxyazetidinone process does not yet have a rating. At this time, there are no reviews or comments for this patent.

If you have personal experience with Stereocontrolled acetoxyazetidinone process, we encourage you to share that experience with our LandOfFree.com community. Your opinion is very important and Stereocontrolled acetoxyazetidinone process will most certainly appreciate the feedback.

Rate now

Comments { 0 }

Profile ID: LFUS-PAI-O-857236