Synthesis of acylated benzothiophenes

Details Synthesis of acylated benzothiophenes Synthesis of acylated benzothiophenes

1981-12-16

1983-04-19

Raymond, Richard

Organic compounds -- part of the class 532-570 series

Organic compounds

Heterocyclic carbon compounds containing a hetero ring...

2603303, 544146, 548525, 549 51, C07D33364

Patent

active

043806350

ABSTRACT:
A group of 6-hydroxy-2-(4-hydroxyphenyl)-3-[4-(2-aminoethoxy)benzoyl]benzo[b]thiophen es are prepared by acylation of a methyl-protected starting compound followed by demethylation in a single reaction mixture.

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