Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Heterocyclic carbon compounds containing a hetero ring...
Patent
1996-02-20
1997-12-02
Grumbling, Matthew V.
Drug, bio-affecting and body treating compositions
Designated organic active ingredient containing
Heterocyclic carbon compounds containing a hetero ring...
5142382, 5142388, 514317, 514331, 514424, 544 59, 544158, 546240, 546264, 546312, 548542, A61K 3154, A61K 31535, C07D40102, C07D24912
Patent
active
056936397
ABSTRACT:
Compounds of formula I ##STR1## wherein R.sup.1, R.sup.2, R.sup.3, R.sup.4, R.sup.5 and A-B have any of the meanings given in the specification, and their pharmaceutically acceptable salts are useful in the treatment of urinery incontinence. Also disclosed are pharmaceutical compositions, processes for preparing the compounds of formula I and intermediates.
REFERENCES:
patent: 3291837 (1966-12-01), Goldberg et al.
patent: 3365485 (1968-01-01), Bell
patent: 3468878 (1969-09-01), Bell
patent: 3661917 (1972-05-01), Kaiser et al.
patent: 3662071 (1972-05-01), Langkammerer
patent: 3715375 (1973-02-01), Shen et al.
patent: 3885047 (1975-05-01), Seidehamel et al.
patent: 3998890 (1976-12-01), Glen
patent: 4239776 (1980-12-01), Glen
patent: 4282218 (1981-08-01), Glen et al.
patent: 4330542 (1982-05-01), Descamps et al.
patent: 4386080 (1983-05-01), Crossley et al.
patent: 4535092 (1985-08-01), Hughes
patent: 4636505 (1987-01-01), Tucker
patent: 4845119 (1989-07-01), Hughes et al.
patent: 4873329 (1989-10-01), Hughes et al.
patent: 4880839 (1989-11-01), Tucker
patent: 5032592 (1991-07-01), Hughes et al.
patent: 5266589 (1993-11-01), Van Dasler et al.
patent: 5272163 (1993-12-01), Russell et al.
patent: 5403930 (1995-04-01), Agback et al.
patent: 5474999 (1995-12-01), Russell et al.
R Bayles et al., "The Smiles rearrangement of 2-aryloxy-2-methylpropanamides. Synthesis of N-aryl-2-hydroxy-2-methylpropanamides" Synthesis. (1977), 31-33.
G Edwards et al., "Structure-activity relationships of potassium channel openers", Trends in Pharmacological Sciences. (1990), 11, 417-442.
B. Delfort, et al. "Ethynyl-Terminated Polyethers from New End-Capping Agents: Synthesis and Characterization" Journal of Polymer Science: Part A: Polymer Chemistry (1990), 28 (9), 2451-64.
Sandoz Ltd, Chemical Abstracts vol. 52, No. 5, col. 52:4194 through 52:4195, 1958.
Jackman et al, Chemical Abstracts vol. 55, No. 9, cols. 55:8335 through 55:8338, 1961.
J.J. Morris, et al. "Non-Steroidal Antiandrogens. Design of Novel Compounds Based on an Infrared Study of the Dominant Conformations and Hydrogen-Bonding Properties of a Series of Anilide Antiandrogens" J. Med. Chem. (1991), 34, 447-455.
S. Sarel, et al. "Factors Affecting Base-Induced Rearrangements of .alpha.-Chloro-.alpha.-,.alpha.-diphenylacetamides" Journal of Organic Chemistry (1970), 35(6), 1850-1857.
Jackman, et al. "The Condensation of Some Halogeno-2,4-Disulphamyl-Benzene Derivatives with Basic Reagents" Journal of Pharm. Pharmacol. (1960) , 12, 648-655.
Empfield James Roy
Mayhugh Daniel Ray
Russell Keith
Grumbling Matthew V.
Hohenschutz Liza D.
Zeneca Limited
LandOfFree
Therapeutic heterocyclyl amionosulfonyl phenyl compounds does not yet have a rating. At this time, there are no reviews or comments for this patent.
If you have personal experience with Therapeutic heterocyclyl amionosulfonyl phenyl compounds, we encourage you to share that experience with our LandOfFree.com community. Your opinion is very important and Therapeutic heterocyclyl amionosulfonyl phenyl compounds will most certainly appreciate the feedback.
Profile ID: LFUS-PAI-O-801447