Substituted oxotremorine derivatives

Details Substituted oxotremorine derivatives Substituted oxotremorine derivatives

1996-04-30

1997-06-10

Springer, David B.

Organic compounds -- part of the class 532-570 series

Organic compounds

Heterocyclic carbon compounds containing a hetero ring...

548545, 548550, C07D207277

Patent

active

056377312

ABSTRACT:
This disclosure describes novel substituted oxotremorine derivatives of formula I having nitrogen, oxygen or sulfur groups and the prodrug forms of these derivatives. The compounds have cholinergic activity. Also disclosed are methods for treating diseases of the central nervous system in mammals employing the compounds, pharmaceutical preparations containing the compounds and the processes for the production of the compounds. ##STR1##

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