Substituted benzoate ester prodrug derivatives of 3-hydroxymorph

Details Substituted benzoate ester prodrug derivatives of 3-hydroxymorph Substituted benzoate ester prodrug derivatives of 3-hydroxymorph

1985-05-14

1987-05-26

Daus, Donald G.

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Having -c-, wherein x is chalcogen, bonded directly to...

514282, 514289, 546 39, 546 44, 546 45, 546 46, 546 63, 546 74, A61K 31485, C07D48912, C07D48902, C07D22128

Patent

active

046686851

ABSTRACT:
Substituted benzoate ester prodrug derivatives of 3-hydroxymorphinans are useful as analgesics or narcotic antagonists and provide enhanced bioavailability of 3-hydroxymorphinans from orally administered doses.

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