Phenyl sulfonamide endothelin antagonists

Details Phenyl sulfonamide endothelin antagonists Phenyl sulfonamide endothelin antagonists

1996-01-11

2000-08-22

Powers, Fiona T.

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Having -c-, wherein x is chalcogen, bonded directly to...

514380, 548241, 548243, 548244, 548245, 548246, A61K 31422, A61K 31423, C07D26116, C07D26112

Patent

active

061073202

ABSTRACT:
Compounds of the formula ##STR1## inhibit the activity of endothelin. The symbols are defined as follows: R.sup.1, R.sup.2 and R.sup.3 are each independently

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