Indenoindoles and benzocarbazoles as estrogenic agents

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Heterocyclic carbon compounds containing a hetero ring...

Patent

Rate now

  [ 0.00 ] – not rated yet Voters 0   Comments 0

Details

540602, A61K 3155, C07D40312

Patent

active

061072923

ABSTRACT:
The present invention relates to new substituted benzo[a]carbazoles and indenoindoles which are useful as estrogenic agents, as well as pharmaceutical compositions and methods of treatment utilizing these compounds, having the general structures below. ##STR1##

REFERENCES:
patent: 4656187 (1987-04-01), Black et al.
patent: 4894373 (1990-01-01), Young
patent: 4943572 (1990-07-01), von Angerer
patent: 5023254 (1991-06-01), von Angerer
patent: 5051442 (1991-09-01), Salituro et al.
patent: 5124335 (1992-06-01), Patchett et al.
patent: 5185360 (1993-02-01), Sainbury et al.
patent: 5389641 (1995-02-01), Naka et al.
patent: 5395842 (1995-03-01), Labrie et al.
patent: 5496844 (1996-03-01), Inai et al.
patent: 5534527 (1996-07-01), Black et al.
patent: 5550107 (1996-08-01), Labrie
patent: 5552401 (1996-09-01), Cullinan et al.
patent: 5591753 (1997-01-01), Black et al.
patent: 5646137 (1997-07-01), Black et al.
patent: 5672609 (1997-09-01), Bryant et al.
patent: 5852039 (1998-12-01), Sohda et al.
von Angerer et al., J. Med. Chem. ., vol. 33, No. 9, pp. 2635-2640, (1990).
von Angerer et al., J. Med. Chem., vol. 30, No. 1., pp. 132-136, (1987).
Rackeley, Contemporary Treatment in Cardiovascular Disease, 1, pp. 49-58 (1996).
von Angerer et al., Ann, N.Y. Aca. Sci., pp. 176, 177, 189, (1995).
Oparil "Hypertension in postmenopausal Woman:Pathology and Management" EMBASE 95:283951, (1995).
von Angerer et al., J. Med. Chem. vol. 27, pp. 1439-1447, (1984).
Biberger, J. Steroid Biochem. Molec., vol. 58, No. 1, pp. 31-43 (1996).
Bone, vol. 17, No. 4, (Oct. 1995) 181S-190S.
Von Angerer, J. Med. Chem. (1983), vol. 26 (1), pp. 113-116.
Kauppila et al., Am. J. Obstet. Gynecol., vol. 140, No. 7, (1981), pp. 787-792.
Kauppila et al., Arch. Gynecol. (1983) 234:49-58.
Segall et al., Eur. J. Med. Chem., 30, No. 2, 165-169 (1995).
Klinicheskaya Farmakologiya i Terapiya, (1996), 5 (1), pp. 70-75.
Klinicheskaya Farmakologiya i Terapiya, (1994), 3 (3), pp. 30-39.
Evans, et al., Bone, 17 (4), (Oct. 1995), pp. 181S-190S.

LandOfFree

Say what you really think

Search LandOfFree.com for the USA inventors and patents. Rate them and share your experience with other people.

Rating

Indenoindoles and benzocarbazoles as estrogenic agents does not yet have a rating. At this time, there are no reviews or comments for this patent.

If you have personal experience with Indenoindoles and benzocarbazoles as estrogenic agents, we encourage you to share that experience with our LandOfFree.com community. Your opinion is very important and Indenoindoles and benzocarbazoles as estrogenic agents will most certainly appreciate the feedback.

Rate now

     

Profile ID: LFUS-PAI-O-581292

  Search
All data on this website is collected from public sources. Our data reflects the most accurate information available at the time of publication.