Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Heterocyclic carbon compounds containing a hetero ring...
Patent
1996-03-27
1998-03-31
Bernhardt, Emily
Drug, bio-affecting and body treating compositions
Designated organic active ingredient containing
Heterocyclic carbon compounds containing a hetero ring...
5142358, 514252, 544 60, 544121, 544357, 544360, 544364, A61K 31495, A61K 31535, C07D40106, C07D41314
Patent
active
057339074
ABSTRACT:
Prodrugs of the HIV protease inhibitor L-735,524 are useful in the inhibition of HIV protease, the prevention or treatment of infection by HIV and the treatment of AIDS, either as compounds, pharmaceutically acceptable salts, pharmaceutical composition ingredients, whether or not in combination with other antivirals, immunomodulators, antibiotics or vaccines. Methods of treating ADS and methods of preventing or treating infection by HIV are also described.
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Alexander Jose
Bindra Dilbir
Dorsey Bruce D.
Repta Arnold J.
Vacca Joseph P.
Appollina Mary A.
Bernhardt Emily
Merck & Co. , Inc.
Tribble Jack L.
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