Drug – bio-affecting and body treating compositions – Preparations characterized by special physical form – Particulate form
Patent
1992-08-31
1994-07-19
Lovering, Richard D.
Drug, bio-affecting and body treating compositions
Preparations characterized by special physical form
Particulate form
424461, 4284022, 42840221, 42840222, 514963, A61K 950, A61K 952, B01J 1304
Patent
active
053307674
ABSTRACT:
Microcapsules are advantageously produced with high take-up of a water-soluble drug by preparing a W/O emulsion composed of a water-soluble drug-containing solution as the inner aqueous phase and a polymer-containing solution as the oil phase, dispersing said emulsion in an aqueous phase and subjecting the resulting W/O/W emulsion to an in-water drying, wherein the viscosity of the W/O emulsion used in preparing the W/O/W emulsion is adjusted to about 150 to about 10,000 centipoises.
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Ogawa Yasuaki
Takada Shigeyuki
Yamamoto Masaki
Lovering Richard D.
Takeda Chemical Industries Ltd.
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