Tricyclic compounds as TXA.sub.2 antagonists

Details Tricyclic compounds as TXA.sub.2 antagonists Tricyclic compounds as TXA.sub.2 antagonists

1992-03-23

1993-09-07

Russell, Mark

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Having -c-, wherein x is chalcogen, bonded directly to...

514309, 514310, 514311, 514312, 514313, 514314, 5142242, 514290, 542 51, 542 52, 546 90, 546141, 546142, 546143, 546144, 546147, 546148, 546155, 546156, 546157, 546159, 546160, 546171, 546172, 546174, 546175, 546167, 549 12, 549354, A61K 3147, C07D40112

Patent

active

052429318

ABSTRACT:
Novel Tricyclic compound represented by formula ##STR1## possess a TXA.sub.2 biosynthesis inhibiting act and/or a TXA.sub.2 receptor antagonizing activity, and are expected to have preventive and therapeutic effects on ischemic diseases, cerebro-vascular diseases, etc.

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