Mercaptoacyl aminolactam endopeptidase inhibitors

Details Mercaptoacyl aminolactam endopeptidase inhibitors Mercaptoacyl aminolactam endopeptidase inhibitors

1990-03-09

1991-12-24

Bond, Robert T.

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Heterocyclic carbon compounds containing a hetero ring...

514212, 514213, 5142222, 5142242, 5142288, 5142305, 5142308, 514299, 514301, 514302, 514312, 514327, 514418, 514424, 540454, 540455, 540490, 540488, 540523, 540524, 540527, 546114, 546115, 546112, 546157, 546244, 548550, 548452, 548484, A61K 3155, C07D22310

Patent

active

050753029

ABSTRACT:
Mercaptoacyl aminolactam inhibitors of endopeptidases of the formula ##STR1## wherein Y is -(CHR.sup.5).sub.n (CR.sup.3 R.sup.4)- or -(CR.sup.3 R.sup.4).sub.p X(CR.sup.3 R.sup.4).sub.q -,

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