Cyclic amine compound

Details Cyclic amine compound Cyclic amine compound

2005-04-08

2009-10-13

Kwon, Brian-Yong S (Department: 1614)

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Having -c-, wherein x is chalcogen, bonded directly to...

C514S292000, C546S198000, C546S199000

Reexamination Certificate

active

07601734

ABSTRACT:
An object of the present invention is to provide a cyclic amine compound which has a potent inhibitory effect on the binding of α2C-adrenoceptor and is useful in preventing and treating disorders attributable to α2C-adrenoceptor.The above-described object is solved by the following cyclic amine compound, etc.,wherein X is O, S, SO, SO2or NR2, etc.; R1is a hydrogen atom, a cyano group, a carboxyl group, a C2-C13alkoxycarbonyl group, a carbamoyl group, etc.; Ar1and Ar2are the same or different and each represent an aryl or heteroaryl group which may be substituted by 1 to 3 substituents and so on; ring B is a benzene ring may be substituted by 1 to 3 substituents and so on; n is an integer from 1 to 10; and p and q are the same or different and each represent an integer of 1 or 2.

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International Search Report dated Jun. 7, 2005.

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