4-(substituted cycloalkylmethyl) imidazole-2-thiones,...

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Having -c- – wherein x is chalcogen – bonded directly to...

Reexamination Certificate

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C546S112000, C546S152000, C514S229800, C514S311000

Reexamination Certificate

active

10950376

ABSTRACT:
The compound of the formulawherein the * indicates an asymmetric carbon, is specific to alpha2Badrenergic receptors in preference over alpha2Aand alpha2Cadrenergic receptors, and as such has no or only minimal cardivascular and/or sedatory activity. The compound is useful as medicament in mammals, including humans, for treatment of diseases and or alleviations of conditions which are responsive to treatment by agonists of alpha2Badrenergic receptors.

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