GlyT2 modulators

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Having -c- – wherein x is chalcogen – bonded directly to...

Reexamination Certificate

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Details

C514S586000, C548S568000, C564S027000

Reexamination Certificate

active

10976067

ABSTRACT:
Certain α-, β-, and γ-amino acid derivatives are disclosed as selective GlyT2 inhibitors for the treatment of central nervous system (CNS) conditions such as muscle spasticity, tinnitus, epilepsy and neuropathic pain.

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International Search Report dated Mar. 31, 2005, for corresponding application PCT/US2004/036009.

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