Oxazolidinone derivatives with antibiotic activity

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Having -c- – wherein x is chalcogen – bonded directly to...

Reexamination Certificate

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C514S340000, C546S210000, C546S271400

Reexamination Certificate

active

07141583

ABSTRACT:
Compounds of the formula (I), or a pharmaceutically acceptable salt, or an in-vivo-hydrolysable ester thereof,wherein HET is an N-linked 5-membered heteroaryl ring, optionally substituted on a C atom by an oxo or thioxo group; and/or by 1 or 2 (1–4C)alkyl groups; and/or on an available nitrogen atom by (1–4C)alkyl; or HET is an N-linked 6-membered heteroaryl ring containing up to three nitrogen heteroatoms in total, optionally substituted on a C atom as above;Q is selected from, for example, Q1R2and R3are independently hydrogen or fluoro;T is selected from a range of groups, for example, of formula (TC5)wherein Rc is, for example, R13CO—, R13SO2— or R13CS—;wherein R13is, for example, optionally substituted (1–10C)alkyl or R14C(O)O(1–6C)alkylwherein R14is optionally substituted (1–10C)alkyl; are useful as antibacterial agents; and processes for their manufacture and pharmaceutical compositions containing them are described.

REFERENCES:
patent: 4150029 (1979-04-01), Dostert et al.
patent: 4287351 (1981-09-01), Bourgery et al.
patent: 4340606 (1982-07-01), Fugitt et al.
patent: 4372967 (1983-02-01), Langlois et al.
patent: 4476136 (1984-10-01), Dostert et al.
patent: 4705799 (1987-11-01), Gregory
patent: 4851423 (1989-07-01), Girijavallabhan et al.
patent: 4942183 (1990-07-01), Gregory et al.
patent: 4948801 (1990-08-01), Carlson et al.
patent: 4977173 (1990-12-01), Brittelli et al.
patent: 5164510 (1992-11-01), Brickner
patent: 5182403 (1993-01-01), Brickner
patent: 5225565 (1993-07-01), Brickner
patent: 5231188 (1993-07-01), Brickner
patent: 5247090 (1993-09-01), Brickner
patent: 5272167 (1993-12-01), Girijavallabhan et al.
patent: 5459144 (1995-10-01), Girijavallabhan et al.
patent: 5480899 (1996-01-01), Yano et al.
patent: 5521202 (1996-05-01), Yano et al.
patent: 5523403 (1996-06-01), Barbachyn
patent: 5529998 (1996-06-01), Habich et al.
patent: 5532255 (1996-07-01), Raddatz et al.
patent: 5547950 (1996-08-01), Hutchinson et al.
patent: 5561148 (1996-10-01), Gante et al.
patent: 5574055 (1996-11-01), Borgulya et al.
patent: 5627181 (1997-05-01), Riedl et al.
patent: 5652238 (1997-07-01), Brickner et al.
patent: 5668286 (1997-09-01), Yamada et al.
patent: 5684023 (1997-11-01), Riedl et al.
patent: 5688792 (1997-11-01), Barbachyn et al.
patent: 5698574 (1997-12-01), Riedl et al.
patent: 5700799 (1997-12-01), Hutchinson et al.
patent: 5708169 (1998-01-01), Hester, Jr. et al.
patent: 5719154 (1998-02-01), Tucker et al.
patent: 5736545 (1998-04-01), Gadwood et al.
patent: 5750532 (1998-05-01), Girijavallabhan et al.
patent: 5785976 (1998-07-01), Westesen et al.
patent: 5792765 (1998-08-01), Riedl et al.
patent: 5827857 (1998-10-01), Riedl et al.
patent: 5837870 (1998-11-01), Pearlman et al.
patent: 5843967 (1998-12-01), Riedl et al.
patent: 5861413 (1999-01-01), Habich et al.
patent: 5869659 (1999-02-01), Stolle et al.
patent: 5880118 (1999-03-01), Barbachyn et al.
patent: 5883093 (1999-03-01), Hutchinson et al.
patent: 5910504 (1999-06-01), Hutchinson
patent: 5922708 (1999-07-01), Riedl et al.
patent: 5929083 (1999-07-01), Yoon et al.
patent: 5952324 (1999-09-01), Barbachyn et al.
patent: 5955460 (1999-09-01), Thomas
patent: 5968962 (1999-10-01), Thomas et al.
patent: 5981528 (1999-11-01), Gravestock
patent: 6028090 (2000-02-01), Gante et al.
patent: 6051716 (2000-04-01), Hutchinson et al.
patent: 6069145 (2000-05-01), Betts
patent: 6069160 (2000-05-01), Stolle et al.
patent: 6090820 (2000-07-01), Barbachyn et al.
patent: 6107519 (2000-08-01), Pearlman
patent: 6110936 (2000-08-01), Gravestock
patent: 6124334 (2000-09-01), Hutchinson
patent: 6129940 (2000-10-01), Leadbeater
patent: 6140318 (2000-10-01), Cama et al.
patent: 6194441 (2001-02-01), Roberts et al.
patent: 6271388 (2001-08-01), Yaegashi et al.
patent: 6362191 (2002-03-01), Mills
patent: 6455529 (2002-09-01), Gante et al.
patent: 6462056 (2002-10-01), Bottcher et al.
patent: 2002/0045625 (2002-04-01), Sciotti et al.
patent: 2002/0103186 (2002-08-01), Mehta et al.
patent: 199 01 306 (2000-07-01), None
patent: 199 07 701 (2000-08-01), None
patent: 199 09 785 (2000-09-01), None
patent: 100 14 961 (2001-01-01), None
patent: 100 34 624 (2002-01-01), None
patent: 100 34 625 (2002-01-01), None
patent: 0 127 902 (1984-12-01), None
patent: 0 184 170 (1986-11-01), None
patent: 0 359 418 (1990-03-01), None
patent: 0 609 905 (1994-08-01), None
patent: 0 710 657 (1996-05-01), None
patent: 1 029 854 (2000-08-01), None
patent: 1 130 016 (2001-09-01), None
patent: 2 338 268 (1977-08-01), None
patent: 2 458 547 (1981-01-01), None
patent: 07-309850 (1995-11-01), None
patent: 11-322729 (1999-11-01), None
patent: 2000-136186 (2000-05-01), None
patent: WO 93/09103 (1993-05-01), None
patent: WO 93/23384 (1993-11-01), None
patent: WO 94/01110 (1994-01-01), None
patent: WO 97/06791 (1997-02-01), None
patent: WO 97/10223 (1997-03-01), None
patent: WO 97/14690 (1997-04-01), None
patent: WO 97/23212 (1997-07-01), None
patent: WO 97/31917 (1997-09-01), None
patent: WO 98/01446 (1998-01-01), None
patent: WO 98/01447 (1998-01-01), None
patent: WO 98/07708 (1998-02-01), None
patent: WO 98/54161 (1998-12-01), None
patent: WO 99/02525 (1999-01-01), None
patent: WO 99/03846 (1999-01-01), None
patent: WO 99/10342 (1999-03-01), None
patent: WO 99/12914 (1999-03-01), None
patent: WO 99/24428 (1999-05-01), None
patent: WO 99/25344 (1999-05-01), None
patent: WO 99/29688 (1999-06-01), None
patent: WO 99/32175 (1999-07-01), None
patent: WO 99/33839 (1999-07-01), None
patent: WO 99/37630 (1999-07-01), None
patent: WO 99/37641 (1999-07-01), None
patent: WO 99/37652 (1999-07-01), None
patent: WO 99/40094 (1999-08-01), None
patent: WO 99/41244 (1999-08-01), None
patent: WO 99/43671 (1999-09-01), None
patent: WO 99/59616 (1999-11-01), None
patent: WO 99/62504 (1999-12-01), None
patent: WO 99/63937 (1999-12-01), None
patent: WO 99/64416 (1999-12-01), None
patent: WO 99/64417 (1999-12-01), None
patent: WO 00/03710 (2000-01-01), None
patent: WO 00/10566 (2000-03-01), None
patent: WO 00/21960 (2000-04-01), None
patent: WO 00/27816 (2000-05-01), None
patent: WO 00/27817 (2000-05-01), None
patent: WO 00/27827 (2000-05-01), None
patent: WO 00/29396 (2000-05-01), None
patent: WO 00/29409 (2000-05-01), None
patent: WO 00/32599 (2000-06-01), None
patent: WO 00/41473 (2000-07-01), None
patent: WO 00/44741 (2000-08-01), None
patent: WO 00/45177 (2000-08-01), None
patent: WO 00/62783 (2000-10-01), None
patent: WO 00/73301 (2000-12-01), None
patent: WO 01/40222 (2001-06-01), None
patent: WO 01/40236 (2001-06-01), None
patent: WO 01/42229 (2001-06-01), None
patent: WO 01/42242 (2001-06-01), None
patent: WO 01/44212 (2001-06-01), None
patent: WO 01/46164 (2001-06-01), None
patent: WO 01/46185 (2001-06-01), None
patent: WO 01/47919 (2001-07-01), None
patent: WO 01/58885 (2001-08-01), None
patent: WO 01/74812 (2001-10-01), None
patent: WO 01/80841 (2001-11-01), None
patent: WO 01/81350 (2001-11-01), None
patent: WO 01/94342 (2001-12-01), None
patent: WO 01/98297 (2001-12-01), None
patent: WO 02/02095 (2002-01-01), None
patent: WO 02/15940 (2002-02-01), None
patent: WO 02/18354 (2002-03-01), None
patent: WO 02/20515 (2002-03-01), None
patent: WO 02/32459 (2002-04-01), None
patent: WO 02/32857 (2002-04-01), None
patent: WO 02/48139 (2002-06-01), None
patent: WO 02/50040 (2002-06-01), None
patent: WO 02/050061 (2002-06-01), None
patent: WO 02/051819 (2002-07-01), None
patent: WO 02/056013 (2002-07-01), None
patent: WO 02/059115 (2002-08-01), None
patent: WO 02/059116 (2002-08-01), None
patent: WO 02/080841 (2002-10-01), None
patent: WO 02/081468 (2002-10-01), None
patent: WO 02/081469 (2002-10-01), None
patent: WO 02/081470 (2002-10-01), None
patent: WO 02/096890 (2002-12-01), None
patent: WO 02/096916 (2002-12-01), None
patent: WO 02/096917 (2002-12-01), None
patent: WO 02/096918 (2002-12-01), None
patent: WO 02/102785 (2002-12-01), None
patent: WO 03/000256 (2003-01-01), None
1995-2002 ICAAC (Interscience Congress of Antimicrobial Agents and Chemotherapy) conference abstracts.
Ashtekar, D. et al. Oxazolidinones, a New Class of

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