Peptide having an ability to promote the activation of protein C

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Peptide containing doai

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435 696, 4353201, 435325, 4352523, 530350, 530380, 530381, A61K 3817, A61K 3836, C12N 1512

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060340606

ABSTRACT:
The peptide of the present invention comprises a specific amino acid sequence including at least 118 amino acids and has the ability to promote the activation of protein C by thrombin. The peptide of the present invention can be produced efficiently on a large scale by recombinant DNA techniques. The peptide of the present invention has anticoagulant, platelet aggregation-inhibiting and thrombolytic activities, without exhibiting side effects such as bleeding and anaphylactic shock. Therefore, the peptide of the present invention can be effectively used for the treatment of various circulatory organ diseases, toxemia of pregnancy and the like.

REFERENCES:
patent: 4638050 (1987-01-01), Aoki
patent: 4748156 (1988-05-01), Aoki et al.
patent: 4912207 (1990-03-01), Majerus
patent: 5466668 (1995-11-01), Glaser et al.
patent: 5516659 (1996-05-01), Nii et al.
patent: 5583102 (1996-12-01), Lentz et al.
Cuatrecasas, P., J. Biol. Chem., 245(12) : 3059-3065, 1970.
Salem et al. "Kolabirn & Characterization of Thrombomodulin from Human Placenta" J. Biol. Chemistry v. 259(19) 12246-12251 (Oct. 10, 1984).
Wen, D "Human Thrombomodulin:Complete cDNA Sequence & Chromosome Localization of the Gene" Biochemistry 26:4350-4357 (Jul. 14, 1987) 1986/1987 IBI Catalog "Life on the Edge" vol. II published by International Biotechnologies, Inc. pp. 78-79.
Suzuki et al, The EMBO Journal, 6, No. 7, pp. 1891-1897 (1987).
Wen et al, Biochemistry, 26, pp. 4350-4357 (1987).
Jackman et al, Proc. Natl. Acad. Sci. USA, 83, pp. 8834-8838 (1986).
Hidemi Ishii et al, "Thrombomodulin Is Present in Human Plasma and Urine", J. Clin. Invest. vol. 76, (1985) pp. 2178-2181.
Shinichiro Kurosawa et al., "Proteolytic Formation and Properties of Functional Domains of Thrombomodulin", The Journal of Biological Chemistry, vol. 262, No. 5, (1987) pp. 2206-2212.
Koji Suzuki et al., "Isolation and charaterization of thrombomodulin from bovine lung", Biochimica et Biophysica Acta 882 (1986) pp. 343-352.
Robert W. Jackman et al., "Human thrombomodulin gene is intron depleted: Nucleic acid sequences of the cDNA and gene predict protein structure and suggest sites of regulatory control", Proc. Natl. Acad. Sci. USA, vol. 84 (1987) pp. 6424-6429.
Hiroshi Kusumoto, "Thrombomodulin, A Cofactor of Protein C Activation: Isolation, Characterization and Application for Laboratory Medicine", Mie Medical Journal, vol. 37 No. 1 (1987) pp. 145-172.
D. Wen et al., "Human Thrombomodulin:CDNA Cloning and Primary Structure", Clinical Research, vol. 35, No. 3 (1987) p. 603A.
N.L. Esmon et al., J. Biol. Chem., vol. 257, p. 859 (1982).
C.T. Esmon et al., Proc. Natl. Acad. Sci. USA, vol. 78, p. 2249 (1981).
C.T. Esmon et al., J. Biol. Chem., vol. 257, p. 7944 (1982).
N.L. Esmon et al., J. Biol. Chem., vol. 258, p. 12238 (1983).
H.H. Salem et al., J. Biol. Chem., vol. 259, p. 12246 (1984).
S.Kurosawa et al., Thromb. Res., vol. 37, p. 353 (1985).
Kusumoto et al., Biochemistry, Japan, vol. 56, p. 890 (1984).
Kusumoto et al., Biochemistry, Japan, vol. 57, p. 1102 (1985).

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