Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Having -c- – wherein x is chalcogen – bonded directly to...
Reexamination Certificate
2006-10-24
2006-10-24
Shameem, Golam M. M. (Department: 1626)
Drug, bio-affecting and body treating compositions
Designated organic active ingredient containing
Having -c-, wherein x is chalcogen, bonded directly to...
C548S241000, C548S360100, C549S059000, C514S406000, C514S444000
Reexamination Certificate
active
07125903
ABSTRACT:
The compounds are of the class thienoisoxazolyl- and thienylpyrrazolyl-phenoxy substituted propyl derivatives, useful as D4antagonists. Said compounds are useful for the treatment of medical conditions mediated by inhibition of D4receptor. These conditions comprise, for example, Attention Deficit Hyperactivity Disorder, Obsessive-Compulsive Disorder, Psychoses, Substance Abuse, Substance Dependence, Parkinson's Disease, Parkinsonism, Tardive Diskinesia, Gilles de la Tourette Syndrome, Conduct Disorder, and Oppositional Defiant Disorder. A further aspect of the invention is to provide a pharmaceutical composition, intermediates, and a method of making said class of compounds.
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Fink David M.
Freed Brian S.
Hrib Nicholas J.
Kosley, Jr. Raymond W.
Lee George E.
Aventis Pharmaceuticals Inc.
Kurys Barbara E.
Shameem Golam M. M.
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